Sunday, August 25, 2024
14:00 – 14:30
Opening ceremony
14:30 – 15:30
Plenary Lecture
Electrocatalyzed C-H Activation with Potential
Lutz Ackermann (Georg-August-University Göttingen)
15:30 – 16:15
Coffee break
Chair:
Miroslav Soural
16:15 – 16:45
Blue Danube Senior
Design of Oligothienyl Acenes with Electron Withdrawing Groups as n-type Semiconductors
Martin Putala
16:45 – 17:00
Oral communication 1
Aleš Růžička – The Lightest Metal in Action; Novel Heterocycles, Associates and Clusters of Organolithiums
17:00 – 17:15
Oral communication 2
Sergio Armantia Matheu – Development of Novel Fluorescent Dyes and Their Application as Probes to Study Biological Processes
17:15 – 17:30
Oral communication 3
Petra Sőregi – High density information storage through isotope ratio encoding
17:30 – 17:45
Oral communication 4
Kiryl Vasiutovich – The use of palladium-catalyzed tandem reactions in the synthesis of poly(hetero)cyclic and spirocyclic compounds
17:45 – 18:00
Oral communication 5
Stanislav Kukla – Merck Lecture – Synple, Safe and Sustainable SnAP Synthesis of Saturated N-Heterocycles
18:00 – 20:00
Welcome reception
Monday, August 26, 2024
Chair:
Martin Putala
9:00 – 9:45
Invited Lecture
Modifications of Heterocyclic Nucleobases in Nucleotides and Nucleic Acids for Applications in Chemical Biology
Michal Hocek (Institute of Organic Chemistry and Biochemistry of The CAS)
9:45 – 10:05
Blue Danube Junior
Light-Mediated Nickel Catalysis Enabled by Donor-Acceptor Ligands
Bartholomäus Pieber (Institute of Science and Technology Austria – ISTA)
10:05 – 10:20
Oral communication 6
Ines Kulašić – Visible-light-induced transformations of pyrazolo[1,2-a]pyrazolones
10:20 – 10:35
Oral communication 7
Ivana Weisheitelová – 5-Aryldeazaalloxazine radicals as a new efficient tool in photoreductions
10:35 – 11:00
Coffee break
Chair:
Marko D. Mihovilovic
11:00 – 11:30
Blue Danube Senior
Bioorthogonal Modulation of Photoresponsivity and Vice Versa
Péter Kele (Research Centre for Natural Sciences, Hungary)
11:30 – 11:45
Oral communication 8
Jure Gregorc – Trifluoromethylthiolation of aromatic amino acids: Peptide late-stage functionalization, local hydrophobicity modulation and selective post-oxidation
11:45 – 12:00
Oral communication 9
Grisa Princic – Advanced Reagent for Nucleophilic Fluorination
12:00 – 12:15
Oral communication 10
Antonio Massa – Organocascade reactions of functionalized α-amidosulfones in the asymmetric synthesis of bioactive γ-lactams
12:15 – 12:30
Oral communication 11
Paulo Paioti – Rapid Synthesis of Diverse Heterocyclic C‒N Atropisomers
12:30 – 12:50
Blue Danube Junior
Copper-Catalyzed Synthesis of Vinyl Sulfones and Sulfonamides under Visible Light
Nejc Petek (University of Ljubljana)
12:50 – 14:00
Lunch
13:40 – 14:40
Steering Committee meeting
14:00 – 16:00
Excursion to Chlupáč Anthropological Museum and Minaralogical Museum
16:00 – 18:00
Boat Cruise at Vltava River
19:00 – 21:00
Speakers Dinner
Tuesday, August 27, 2024
Chair:
Péter Kele
9:00 – 9:45
Invited Lecture
Innovation in Reagents and Catalysts. From Fundamentals to Immediate Application
Josep Cornella (Max-Planck-Institut für Kohlenforschung)
9:45 – 10:05
Blue Danube Junior
Catalytic Enantioselective Nucleophilic Desymmetrization at P(V)
Branislav Ferko (Slovak University of Technology)
10:05 – 10:20
Oral communication 12
Rafael Navrátil – Multimetallic Pd- and Ni-Catalyzed C(sp2)–P Cross-Coupling under Aqueous Micellar Conditions
10:20 – 10:35
Oral communication 13
Luka Jedlovčnik – Towards Selective Deuteration of Diazine Carboxamides via Directed Ortho Metalation
10:35 – 11:00
Coffee break
Chair:
Radek Cibulka
11:00 – 11:30
Blue Danube Senior
Weakly interacting heterocyclic motifs as the basis of highly selective inhibitors of underexplored protein kinases
Kamil Paruch (Masaryk University, Brno)
11:30 – 11:45
Oral communication 14
Ondřej Baszczyňski – Phosphorus Self-Immolative Linkers in Prodrug Design
11:45 – 12:00
Oral communication 15
Jan Chasák – Squaramides as Mycobacterial ATP synthase Inhibitors: Synthetic Pathways, Biological Evaluation & Mechanism of Action
12:00 – 12:15
Oral communication 16
Jerneja Kladnik – Synthesis and Evaluation of Novel Fluorescent Probes for Amyloid β Plaques Imaging
12:15 – 12:30
Oral communication 17
Andras Kotschy – Induced proximity by heterocycles: molecular glues and beyond
12:30 – 13:45
Lunch
Chair:
Kamil Paruch
13:45 – 14:05
Blue Danube Junior
Utilization of Conventional Lewis Acids as Bases: Complexes of Carboranes with N-Heterocyclic Carbenes as Catalysts
Jan Vrána (University of Pardubice)
14:05 – 14:20
Oral communication 18
Florian Rudroff – A concurrent cascade towards unsymmetric pyrazines – a hell of a smell
14:20 – 14:35
Oral communication 19
Viktor Iaroshenko – Mechanochemical synthesis of 3-substituted chromones
14:35 – 14:50
Oral communication 20
Nina Biedermann – A solvent-free ultra-fast Wittig olefination – Diels Alder reaction sequence in one-pot under mechanochemical conditions
14:50 – 15:35
Invited Lecture
Chiral Trityls as Versatile Property and Reactivity Platforms
Jérôme Lacour (University of Geneva)
15:35 – 16:05
Coffee break
Chair:
Ondřej Baszczyňski
16:05 – 16:35
Blue Danube Senior
Triggering Formation of Heterocycles Using Biocatalysis
Wolfgang Kroutil (University of Gratz)
16:35 – 16:50
Oral communication 21
Márton Ferenc Szlávik – Synthesis of electron deficient alkenes: useful building blocks for heterocycle formation
16:50 – 17:20
Invited Lecture of the Serbian Representative
Case studies in the chemistry of heterocyclic compounds:
1H-tetrazol-5-amine, pyrazole, pyrimidine and thiophene derivatives
Igor Opsenica (University of Belgrade)
17:20 – 19:00
Poster session
19:30 – 23:00
Conference dinner
Wednesday, August 28, 2024
Chair:
Wolfgang Kroutil
9:00 – 9:45
Invited Lecture
Biomimetic Spirocyclizations for the Synthesis of Indole Alkaloids
Romano Orru (Maastricht University)
9:45 – 10:05
Blue Danube Junior
From Monoterpene Indole Alkaloids to Thianthrenium Salts: A Bioinspired Journey in Organic Synthesis
Szilárd Varga (Research Centre for Natural Sciences, Hungary)
10:05 – 10:20
Oral communication 22
Peter Gabko – Concise stereoselective synthesis of 5-substituted 1,2-dihydroxyindolizidines
and -pyrrolizidines related to natural alkaloids
10:20 – 10:35
Oral communication 23
Raju Hazra – Total Synthesis of the Cryptic Secondary Metabolites Acybolins
10:35 – 11:00
Coffee break
Chair:
Martin Kotora
11:00 – 11:30
Blue Danube Senior
From Lignocellulosic Biomass to Vanillin and Cellulose Hydrogels
Jernej Iskra (University of Ljubljana)
11:30 – 11:45
Oral communication 24
Wim Dehaen – New efficient methods for the synthesis of 1,2,3-triazoles
11:45 – 12:00
Oral communication 25
Sándor Balázs Király – Preparation of bridged- and spirocyclic O,N-heterocycles using domino reactions
12:00 – 12:15
Oral communication 26
Marko D. Mihovilovic – Employing Heterocycles for Quantification and as Redox-Mediators
in Laccase-Catalyzed Starch Oxidation
Closing Remarks